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Target-based Services

Steroid Endocrinology

Aromatase inhibitors

  • In vitro (PDF)
  • In vivo (PDF)
  • Selectivity (ex vivo) (PDF)

P450 17 inhibitors

  • In vitro (PDF)
  • Selectivity (in vitro) (PDF)

5-alpha-reductase Inhibitors

  • In vitro (PDF)
  • In vivo (PDF)

GnRH agonists/antagonists

  • In vitro (PDF)
  • In vivo (PDF)
  • Pre-selection (PDF)
  • PK/PD relationship (PDF)

 

Metabolic syndrome

Diabetes type II

  • In vitro GLP-1 receptor assay (PDF)
  • In vivo rat diabetes model (PDF)